TYPE OF COURSE UNIT	Compulsory Course
LEVEL OF COURSE UNIT	Bachelor's Degree
YEAR OF STUDY	3
SEMESTER	Fifth Term (Fall)
NUMBER OF ECTS CREDITS ALLOCATED	4
NAME OF LECTURER(S)	Professor Hakkı Erdoğan
LEARNING OUTCOMES OF THE COURSE UNIT	At the end of this course, the students; 1) Drug design and its steps, 2) Methods ort he optimization of lead compound by molecular modification techniques, 3) The effect of physicochemical properties of drugs and drug-receptor interactions, 4) Biotransformation, 5) General anesthetics, sedatives and hypnotics, tranquilizers, neuroleptics, anticonvulsant drugs, CNS-acting muscle relaxant drugs, and analgesic drugs.
MODE OF DELIVERY	Face to face
PRE-REQUISITES OF THE COURSE	No
RECOMMENDED OPTIONAL PROGRAMME COMPONENT	None
COURSE DEFINITION	Introduction to pharmaceutical chemistry and basic concepts, biotransformations, central nervous system drugs, general anesthetics, sedatif-hypnotices, tranquilizers, neuroleptics, central acting spasmolytics, anticonvulsants, antidepressants, local anesthetics, non-steroidal antiinflammatory drugs, narcotic analgesics.
COURSE CONTENTS	WEEK TOPICS 1st Week Introduction to pharmaceutical chemistry and basic concepts 2nd Week Introduction to pharmaceutical chemistry and basic concepts 3rd Week Introduction to pharmaceutical chemistry and basic concepts 4th Week Drug biotransformation 5th Week Central System drugs, general anaesthetics 6th Week Sedatives and hypnotics 7th Week Midterm-exam 8th Week Tranquülizers 9th Week Neuroleptics / Local anaesthetic 10th Week Antidepressants, antiepileptics / analeptics 11th Week Anti-Alzheimer drugs, antiparkinsons and central acting spasmolytics 12th Week Narcotic analgesics 13th Week Analgesics 14th Week Analgesics
RECOMENDED OR REQUIRED READING	1. Akgün, H., Balkan, A., Bilgin, A.A., Çalış, Ü., Dalkara, S., Erdoğan, H., Erol Demir, D., Ertan, M., Gökhan, N., Özkanlı, F., Palaska, E., Saraç, S. Şafak, C., Tozkoparan. B.: Farmasötik Kimya, Ankara, 2019. 2. Foye?s Principles of Medicinal Chemistry, Lemke and Williams, 7th ed, Lippincott Williams &Wilkins, Kluwers Philadelphia, 2013. 3. Thomas, G., Fundamentals of Medicinal Chemistry, Wiley, 2003. 4. Patrick, G.L., An Introduction to Medicinal Chemistry, Oxford University Press, Oxford, 1999.
PLANNED LEARNING ACTIVITIES AND TEACHING METHODS	Lecture,Questions/Answers,Discussion
ASSESSMENT METHODS AND CRITERIA	Quantity Percentage(%) Mid-term 1 40 Total(%) 40 Contribution of In-term Studies to Overall Grade(%) 40 Contribution of Final Examination to Overall Grade(%) 60 Total(%) 100
ECTS WORKLOAD	Activities Number Hours Workload Midterm exam 1 1 1 Preparation for Quiz 0 0 0 Individual or group work 14 3 42 Preparation for Final exam 1 20 20 Course hours 14 3 42 Preparation for Midterm exam 1 12 12 Laboratory (including preparation) 0 0 0 Final exam 1 2 2 Homework 0 0 0 Total Workload 119 Total Workload / 30 3,96 ECTS Credits of the Course 4
LANGUAGE OF INSTRUCTION	Turkish
WORK PLACEMENT(S)	No